Thermopsidine

Thermopsidine (CC4) is a selective partial agonist at α4β2/α6β2 nAChR with EC50 values of 2.2 μM target α4β2[1].

Product Specifications

CAS Number

[492-02-4]

Product Name Alternative

CC4

UNSPSC

12352005

Hazard Statement

H315-H319-H320

Target

NAChR

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/thermopsidine.html

Smiles

[H][C@@]12CN3C([C@@](C2)([H])CN(C1)CCN4C[C@](C5)([H])C(N6C[C@]5([H])C4)=CC=CC6=O)=CC=CC3=O

Molecular Formula

C24H30N4O2

Molecular Weight

406.52

Precautions

P264-P280-P302+P352-P305+P351+P338-P362

References & Citations

[1]Mariaelvina Sala, et al. CC4, a dimer of cytisine, is a selective partial agonist at α4β2/α6β2 nAChR with improved selectivity for tobacco smoking cessation. Br J Pharmacol. 2013 Feb;168 (4) :835-49.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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