GW809897X
GW809897X is a dual inhibitor of Fluc and VEGFR with IC50 of 0.58 μM and 65 nM, respectively. GW809897X is a protein kinase inhibitor across ATP-dependent and -independent luciferases with potential impact on Fluc reporter assays[1].
Product Specifications
CAS Number
579515-94-9
UNSPSC
12352005
Target
VEGFR
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/gw809897x.html
Solubility
10 mM in DMSO
Smiles
CN(C1=CC=C(NC(NC2=C(Cl)C=CC=C2Cl)=O)C=C1)C3=NC(NC4=CC(C[S+]([O-])(C)=O)=CC=C4)=NC=C3
Molecular Formula
C26H24Cl2N6O3S
Molecular Weight
571.48
References & Citations
[1]Dranchak P, et al. Profile of the GSK published protein kinase inhibitor set across ATP-dependent and-independent luciferases: implications for reporter-gene assays. PLoS One. 2013;8 (3) :e57888.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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