Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

GR-73632

GR-73632 is a novel tachykinin neurokinin 1 (NK-1) receptor agonist[1]. GR-73632 acts directly on the peripheral terminals of primary sensory neurons through NK1 receptor which convey itch signals[2].

Product Specifications

CAS Number

133156-06-6

UNSPSC

12352209

Target

Neurokinin Receptor

Type

Peptides

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Neurological Disease; Endocrinology

Assay Protocol

https://www.medchemexpress.com/gr-73632.html

Purity

99.93

Solubility

DMSO : ≥ 100 mg/mL|H2O : 1 mg/mL (ultrasonic)

Smiles

NCCCCC(N[C@@H](CC1=CC=CC=C1)C(N[C@@H](CC2=CC=CC=C2)C(N3[C@@H](CCC3)C(N([C@@H](CC(C)C)C(N[C@H](C(N)=O)CCSC)=O)C)=O)=O)=O)=O

Molecular Formula

C40H59N7O6S

Molecular Weight

766.00

References & Citations

[1]Sakurada C, et al. Spinal actions of GR73632, a novel tachykinin NK1 receptor agonist. Peptides. 1999;20 (2) :301-4.|[2]Costantini VJ, et al. The NK1 receptor antagonist aprepitant attenuates NK1 agonist-induced scratching behaviour in the gerbil after intra-dermal, topical or oral administration. Exp Dermatol. 2015 Apr;24 (4) :312-4.

Shipping Conditions

Blue Ice

Storage Conditions

-80°C, 2 years; -20°C, 1 year (Powder, sealed storage, away from moisture and light, under nitrogen)

Scientific Category

Peptides

Clinical Information

No Development Reported

Isoform

NK1R

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-01 0.02 mg (E-Coli)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details
Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-02 0.1 mg (E-Coli)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details
Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-03 0.02 mg (Yeast)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details
Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-04 0.1 mg (Yeast)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details
Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-05 0.02 mg (Baculovirus)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details
Recombinant Mouse Cathepsin J (Ctsj)
MBS1458165-06 0.02 mg (Mammalian-Cell)

Recombinant Mouse Cathepsin J (Ctsj)

Sign In for Pricing
View Details