Cyt-PTPε Inhibitor-1
Cyt-PTPε Inhibitor-1 is a potent cytosolic protein tyrosine phosphatase epsilon (cyt-PTPε) inhibitor, binds to the catalytic domain of cyt-PTPε, blocks c-Src activation (dephosphorylation of c-Src), and exhibits anti-osteoclastic activity[1].
Product Specifications
CAS Number
[428478-94-8]
UNSPSC
12352005
Target
Phosphatase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/cyt-ptp-epsilon-inhibitor-1.html
Purity
98.05
Solubility
10 mM in DMSO
Smiles
O=C(NC1=CC=C(C)C=C1)NC2=NN=C(COC3=CC=C(C)C=C3C)S2
Molecular Formula
C19H20N4O2S
Molecular Weight
368.46
References & Citations
[1]Ku B, et al. Identification of N- (5- (phenoxymethyl) -1,3,4-thiadiazol-2-yl) acetamide derivatives as novel protein tyrosine phosphatase epsilon inhibitors exhibiting anti-osteoclastic activity. ioorg Med Chem. 2018 Oct 1;26 (18) :5204-5211.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
More Discoveries
Explore Other Products
Browse additional items from our catalog
K3632502 1.0 µg DNA
Unc80 sgRNA CRISPR Lentivector (Mouse) (Target 1)
Sign In for Pricing
View Details 
VAng-Cr4396-inquire Inquire
Recombinant HAdV-7 PTP Protein (aa 1-640)
Sign In for Pricing
View Details 
MBS6440140-01 0.1 mL
TCF4 (Transcription Factor 4, E2-2, ITF2, PTHS, SEF2, ITF-2, SEF-2, TCF-4, SEF2-1, SEF2-1A, SEF2-1B, bHLHb19) (HRP)
Sign In for Pricing
View Details MBS6440140-02 5x 0.1 mL
TCF4 (Transcription Factor 4, E2-2, ITF2, PTHS, SEF2, ITF-2, SEF-2, TCF-4, SEF2-1, SEF2-1A, SEF2-1B, bHLHb19) (HRP)
Sign In for Pricing
View Details