EHMT2-IN-1
EHMT2-IN-1 is a potent EHMT inhibitor, with IC50s of all [1].
Product Specifications
CAS Number
[2230849-55-3]
UNSPSC
12352005
Target
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ehmt2-in-1.html
Purity
99.85
Solubility
DMSO : 55 mg/mL (ultrasonic)
Smiles
COC1=C(N2N=CC(CNC)=C2)C=C(NC3=NC(NC)=CC(C)=N3)C=C1
Molecular Formula
C18H23N7O
Molecular Weight
353.42
References & Citations
[1]John Emmerson Campbell, et al. Amine-substituted heterocyclic compounds as ehmt2 inhibitors and methods of use thereof. WO2018118842A1
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
EHMT1/GLP/KMT1D; EHMT2/G9a/KMT1C
Available Sizes
Curated Selection
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