[Lys5, MeLeu9, Nle10]-NKA (4-10)
[Lys5, MeLeu9, Nle10]-NKA (4-10) is a highly selective and potent NK2 receptor agonist, with an IC50 of 6.1 nM[1].
Product Specifications
CAS Number
137565-28-7
UNSPSC
12352209
Target
Neurokinin Receptor
Type
Peptides
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/lys5-meleu9-nle10-nka-4-10.html
Solubility
H2O
Smiles
[DKFVG{N(Me)Leu}{Nle}-NH2]
Molecular Formula
C39H65N9O9
Molecular Weight
803.99
References & Citations
[1]G Chassaing, et al. Selective agonists of NK-2 binding sites highly active on rat portal vein (NK-3 bioassay) . Neuropeptides. 1991 Jun;19 (2) :91-5.|[2]M A Matuszek, et al. An investigation of tachykinin NK2 receptor subtypes in the rat. Eur J Pharmacol. 1998 Jul 3;352 (1) :103-9.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog