BRS-3 receptor agonist-2

BRS-3 receptor agonist-2 (compound 2) is a potent BRS-3 receptor agonist, with an EC50 of 2.5 nM for mouse BRS-3 receptor[1].

Product Specifications

CAS Number

[1021937-07-4]

UNSPSC

12352005

Target

Bombesin Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/brs-3-receptor-agonist-2.html

Solubility

10 mM in DMSO

Smiles

CCC(C)(CC1=CN=C(N1)CCC2=CC=C(C3=NC=CC=C3)C=C2)C

Molecular Formula

C22H27N3

Molecular Weight

333.47

References & Citations

[1]Chobanian HR, et, al. Discovery of MK-7725, A Potent, Selective Bombesin Receptor Subtype-3 Agonist for the Treatment of Obesity. ACS Med Chem Lett. 2012 Jan 21;3 (3) :252-6.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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