(R) -GSK 2830371
(R) -GSK 2830371 is the R-enantiomer of GSK 2830371. GSK 2830371 is a highly selective Wip1 phosphatase inhibitor with IC50 of 6 nM[1].
Product Specifications
CAS Number
2743427-27-0
UNSPSC
12352005
Target
Phosphatase
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/r-gsk-2830371.html
Purity
99.69
Solubility
DMSO : 200 mg/mL (ultrasonic)
Smiles
ClC1=CN=C(C)C(NCC2=CC=C(C(N[C@H](CC3CCCC3)C(NC4CC4)=O)=O)S2)=C1
Molecular Formula
C23H29ClN4O2S
Molecular Weight
461.02
References & Citations
[1]Gilmartin AG, et al. Allosteric Wip1 phosphatase inhibition through flap-subdomain interaction. Nat Chem Biol. 2014 Mar;10 (3) :181-7.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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