(Rac) -WRC-0571
(Rac) -WRC-0571 is a highly potent, orally active and selective, non-xanthine antagonist of A1 adenosine receptors. (Rac) -WRC-0571 inhibits [3H]-N6-cyclohexyladenosine (CHA) binding to guinea pig A1-receptors with a Ki value of 1.1 nM[1].
Product Specifications
CAS Number
501667-77-2
UNSPSC
12352005
Target
Adenosine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/rac-wrc-0571.html
Smiles
OC1C2CC(C1)C(NC3=C4N=C(N(C4=NC=N3)C)N(C(C)C)C)C2
Molecular Formula
C17H26N6O
Molecular Weight
330.43
References & Citations
[1]P L Martin, et al. Characterization of 8- (N-methylisopropyl) amino-N6- (5'-endohydroxy- endonorbornyl) -9-methyladenine (WRC-0571), a highly potent and selective, non-xanthine antagonist of A1 adenosine receptors. J Pharmacol Exp Ther. 1996 Feb;276 (2) :490-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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