DCSM06-05
DCSM06-05 is a potent SMARCA2-BRD inhibitor with an IC50 value of 9 µM, a Kd value of 22.4 µM[1].
Product Specifications
CAS Number
880811-10-9
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/dcsm06-05.html
Smiles
COC1=CC(CNCC2=CC=CC=N2)=CC=C1OCC3=C(F)C=CC=C3
Molecular Formula
C21H21FN2O2
Molecular Weight
352.40
References & Citations
[1]Lu T, et al. Identification of small molecule inhibitors targeting the SMARCA2 bromodomain from a high-throughput screening assay. Acta Pharmacol Sin. 2018 Sep;39 (9) :1544-1552.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
Brd
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