JG-2016
Product Specifications
UNSPSC Description
JG-2016 is a potent inhibitor of histone acetyltransferase 1 (HAT1), with an IC50 of 14.8 μM in the HAT1 acetylation assays[1].
Target Antigen
Histone Acetyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/jg-2016.html
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
O=C(N1)N=C2N(CCOCC(C)C)C3=CC(CC)=C(Cl)C=C3N=C2C1=O
Molecular Weight
376.84
References & Citations
[1]Joshua James GRUBER, et al. Modulators of histone acetyltransferase 1 and methods of treatment thereof. Patent, WO2022272313A1.
Shipping Conditions
Room Temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-154944/JG-2016-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-154944/JG-2016-SDS-MedChemExpress.pdf
Clinical Information
No Development Reported
CAS Number
2887480-87-5
Available Sizes
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
Canine keyhole limpet hemocyanin, KLH IgM antibody (KLH IgM Ab) ELISA Kit
Canine keyhole limpet hemocyanin, KLH IgM antibody (KLH IgM Ab) ELISA Kit
Canine keyhole limpet hemocyanin, KLH IgM antibody (KLH IgM Ab) ELISA Kit
Canine keyhole limpet hemocyanin, KLH IgM antibody (KLH IgM Ab) ELISA Kit