P300-IN-4
P300-IN-4 (compound 6) is a (p300) inhibitor with the IC50 of 12.2 μM.
Product Specifications
UNSPSC
12352005
Target
Histone Acetyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/p300-in-4.html
Smiles
CNC(C[C@@H](NC(C1=CC=C2C(N(NC2=C1)CC(C(O)=O)CC3=CC=C(C=C3)Cl)=O)=O)CC4=CC=C(C=C4)I)=O
Molecular Formula
C29H28ClIN4O5
Molecular Weight
674.91
References & Citations
[1]Suo Y, et al. Discovery Small-Molecule p300 Inhibitors Derived from a Newly Developed Indazolone-Focused DNA-Encoded Library. Bioconjug Chem. 2024;35 (8) :1251-1257.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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