22-Thiocyanatosalvinorin A
22-Thiocyanatosalvinorin A (RB-64) is a potent and selective kappa-opioid receptor agonist with an EC50 of 0.077 nM[1].
Product Specifications
CAS Number
1174223-49-4
Product Name Alternative
RB-64
UNSPSC
12352211
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/22-thiocyanatosalvinorin-a.html
Smiles
C[C@@]12[C@]3([H])[C@]([C@@H](C[C@@H](C3=O)OC(CSC#N)=O)C(OC)=O)(CC[C@@]1([H])C(O[C@H](C4=COC=C4)C2)=O)C
Molecular Formula
C24H27NO8S
Molecular Weight
489.54
References & Citations
[1]Yan F, et al. Structure-based design, synthesis, and biochemical and pharmacological characterization of novel salvinorin A analogues as active state probes of the kappa-opioid receptor. Biochemistry. 2009 Jul 28;48 (29) :6898-908.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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