CCK-A receptor inhibitor 1
CCK-A receptor inhibitor 1 is a cholecystokinin A (CCK-A) receptor inhibitor with a binging IC50 of 340 nM.
Product Specifications
CAS Number
[137004-80-9]
UNSPSC
12352005
Target
Cholecystokinin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease; Endocrinology
Assay Protocol
https://www.medchemexpress.com/Pentanoic_acid,_5-[_3-methoxypropyl_pentylamino]-4-[_2-naphthalenylsulfonyl_methyl]-5-oxo-.html
Solubility
10 mM in DMSO
Smiles
O=C(O)CCC(CS(=O)(C1=CC=C2C=CC=CC2=C1)=O)C(N(CCCOC)CCCCC)=O
Molecular Formula
C25H35NO6S
Molecular Weight
477.61
References & Citations
[1]Ajisawa Y, et al. [Studies on the synthesis of cholecystokinin A receptor antagonists. III. Synthesis and cholecystokinin A receptor inhibitory activities of naphthyl sulfone derivatives]. Yakugaku Zasshi. 1996 Aug;116 (8) :647-56.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CCKAR
Available Sizes
Curated Selection
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