5-HT2 antagonist 1
5-HT2 antagonist 1 is a potent antagonist of 5-HT2 receptor, with weak α1 adrenoceptor blocking activity.
Product Specifications
CAS Number
191592-09-3
UNSPSC
12352005
Target
5-HT Receptor; Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Cardiovascular Disease; Endocrinology
Assay Protocol
https://www.medchemexpress.com/Pyrrolo[3,2-c]azepin-4_1H_-one,_5-[3-[4-_4-fluorophenyl_-1-piperazinyl]propyl]-5,6,7,8-tetrahydro-8-hydroxy-1-methyl-.html
Solubility
10 mM in DMSO
Smiles
O=C1N(CCCN2CCN(C3=CC=C(F)C=C3)CC2)CCC(O)C4=C1C=CN4C
Molecular Formula
C22H29FN4O2
Molecular Weight
400.49
References & Citations
[1]Mizuno A, et al. Synthesis and serotonin 2 (5-HT2) receptor antagonist activity of 5-aminoalkyl-substituted pyrrolo[3,2-c]azepines and related compounds. Chem Pharm Bull (Tokyo) . 2000 May;48 (5) :623-35.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
α-1 microglobulin
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