5-HT2A antagonist 1
5-HT2A antagonist 1 is a 5-HT2A antagonist extracted from patent US5728835A and JP 1007727. 5-HT2A antagonist 1 may be useful in treatment of gastrointestinal disorders circulatory disorders.
Product Specifications
CAS Number
204643-75-4
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/Benzamide,_4-amino-N-[2-_4-benzoyl-1-piperidinyl_ethyl]-N-3-pyridinyl-.html
Solubility
10 mM in DMSO
Smiles
O=C(N(CCN1CCC(C(C2=CC=CC=C2)=O)CC1)C3=CC=CN=C3)C4=CC=C(N)C=C4
Molecular Formula
C26H28N4O2
Molecular Weight
428.53
References & Citations
[1]Aoki Tsuyoshi, et al. Substituted cyclic amine compound, production process thereof and pharmaceutical composition for circulatory organ use containing the same. US5728835A|[2]Preparation of 3-pyridylamines as 5-HT2 receptor antagonists for treatment of circulatory disorders
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT2 Receptor; α-1 microglobulin
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