Cicloprolol (hydrochloride)

Cicloprolol is a partial β 1-adrenoceptor agonist .

Product Specifications

CAS Number

[63686-79-3]

UNSPSC

12352005

Target

Adrenergic Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Cardiovascular Disease; Endocrinology

Assay Protocol

https://www.medchemexpress.com/Cicloprolol_(hydrochloride).html

Solubility

10 mM in DMSO

Smiles

OC(CNC(C)C)COC1=CC=C(OCCOCC2CC2)C=C1.[H]Cl

Molecular Formula

C18H30ClNO4

Molecular Weight

359.89

References & Citations

[1]Weber S, et al. Pharmacodynamic without pharmacokinetic interaction between cicloprolol, a partial beta 1-adrenoceptor agonist, and digoxin in healthy subjects. Br J Clin Pharmacol. 1990 Sep;30 (3) :411-6|[2]Cocco G, et al. An evaluation of the safety of the beta-modulator cicloprolol in chronic heart failure. Clin Cardiol. 1992 Jan;15 (1) :38-42.