(-) -GSK598809
(-) -GSK598809 ((1S,5R) -GSK598809) is an isomer of GSK598809. GSK598809 is a potent and selective dopamine D3 Receptor (DRD3) antagonist.
Product Specifications
CAS Number
863680-46-0
Product Name Alternative
(1S,5R) -GSK598809
UNSPSC
12352005
Hazard Statement
H315-H319
Target
Dopamine Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/1s-5r-gsk598809.html
Solubility
10 mM in DMSO
Smiles
CC1=C(C2=NN=C(SCCCN3C[C@@]4(C5=CC=C(C(F)(F)F)C=C5F)C[C@@]4([H])C3)N2C)OC=N1
Molecular Formula
C22H23F4N5OS
Molecular Weight
481.51
Precautions
P264-P280-P302+P352-P305+P351+P338-P362+P364
References & Citations
[1]Appel NM, et al. Dopamine D3 Receptor Antagonist (GSK598809) Potentiates the Hypertensive Effects of Cocaine in Conscious, Freely-Moving Dogs. J Pharmacol Exp Ther. 2015 Sep;354 (3) :484-92.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
D3 Receptor
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