RWJ-51204

RWJ-51204 is a partial agonist of GABA (A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA (A) receptors.

Product Specifications

CAS Number

[205701-85-5]

UNSPSC

12352005

Target

GABA Receptor

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/RWJ-51204.html

Solubility

10 mM in DMSO

Smiles

O=C(C1=C2N(COCC)C3=CC(F)=CC=C3N2CCC1=O)NC4=CC=CC=C4F

Molecular Formula

C21H19F2N3O3

Molecular Weight

399.39

References & Citations

[1]Dubinsky B, et al. 5-ethoxymethyl-7-fluoro-3-oxo-1,2,3,5-tetrahydrobenzo[4,5]imidazo[1,2a]pyridine-4-N- (2-fluorophenyl) carboxamide (RWJ-51204), a new nonbenzodiazepine anxiolytic. J Pharmacol Exp Ther. 2002 Nov;303 (2) :777-90.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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