RWJ-51204
RWJ-51204 is a partial agonist of GABA (A) receptor, with Ki of 0.2-2 nM to the benzodiazepine site on GABA (A) receptors.
Product Specifications
CAS Number
[205701-85-5]
UNSPSC
12352005
Target
GABA Receptor
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/RWJ-51204.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=C2N(COCC)C3=CC(F)=CC=C3N2CCC1=O)NC4=CC=CC=C4F
Molecular Formula
C21H19F2N3O3
Molecular Weight
399.39
References & Citations
[1]Dubinsky B, et al. 5-ethoxymethyl-7-fluoro-3-oxo-1,2,3,5-tetrahydrobenzo[4,5]imidazo[1,2a]pyridine-4-N- (2-fluorophenyl) carboxamide (RWJ-51204), a new nonbenzodiazepine anxiolytic. J Pharmacol Exp Ther. 2002 Nov;303 (2) :777-90.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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