MAChR-IN-1
MAChR-IN-1 is a potent muscarinic cholinergic receptor (mAChR) antagonist, with an IC50 of 17 nM[1].
Product Specifications
CAS Number
[119391-56-9]
UNSPSC
12352005
Hazard Statement
H315-H319
Target
MAChR
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mAChR-IN-1.html
Purity
99.78
Solubility
DMSO : ≥ 52 mg/mL
Smiles
O=C(C(C1CCN(CC2=CC=C(I)C=C2)CC1)(C3=CC=CC=C3)CC4)NC4=O
Molecular Formula
C23H25IN2O2
Molecular Weight
488.36
Precautions
P264-P280-P302+P352-P305+P351+P338-P362+P364
References & Citations
[1]Wilson AA, et al. Synthesis and biological evaluation of [125I]- and [123I]-4-iododexetimide, a potent muscarinic cholinergic receptor antagonist. J Med Chem. 1989 May;32 (5) :1057-62.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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