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Desformylflustrabromine hydrochloride

Product Specifications

UNSPSC Description

Desformylflustrabromine hydrochloride is a selective agonist of α4β2 neuronal nicotinic acetylcholine receptor (nAChR) with a pEC50 of 6.48.

Target Antigen

nAChR

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel;Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/Desformylflustrabromine_hydrochloride.html

Purity

99.77

Solubility

DMSO : ≥ 105 mg/mL|H2O : 5 mg/mL (ultrasonic)

Smiles

CNCCC1=C(C(C)(C)C=C)NC2=CC(Br)=CC=C12.[H]Cl

Molecular Weight

357.72

References & Citations

[1]Nadezhda German, et al. Deconstruction of the α4β2 Nicotinic Acetylchloine (nACh) Receptor Positive Allosteric Modulator des-Formylflustrabromine (dFBr). J Med Chem. 2011 Oct 27;54(20):7259-67.|[2]Weltzin MM, et al. Desformylflustrabromine Modulates α4β2 Neuronal Nicotinic Acetylcholine Receptor High- and Low-Sensitivity Isoforms at Allosteric Clefts Containing the β2 Subunit. J Pharmacol Exp Ther. 2015 Aug;354(2):184-94.

Shipping Conditions

Room Temperature

Storage Conditions

4°C (Powder, sealed storage, away from moisture)

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-107675/Desformylflustrabromine-hydrochloride-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-107675/Desformylflustrabromine-hydrochloride-SDS-MedChemExpress.pdf

Clinical Information

No Development Reported

CAS Number

951322-11-5

Available Sizes

Curated Selection

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