Glucagon receptor antagonist-1
Glucagon receptor antagonist-1 is a highly potent glucagon receptor antagonist.
Product Specifications
CAS Number
[503559-84-0]
UNSPSC
12352005
Target
GCGR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/glucagon-receptor-antagonists-1.html
Purity
98.65
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
FC1=CC=C(C2=C(/C=C/C)C(C(C)C)=NC(C(C)C)=C2C(C)O)C(OCC3=CC=CC=C3)=C1
Molecular Formula
C29H34FNO2
Molecular Weight
447.58
References & Citations
[1]Ladouceur, Gaetan H. et al. Integration of optimized substituent patterns to produce highly potent 4-aryl-pyridine glucagon receptor antagonists. Bioorganic & Medicinal Chemistry Letters (2002), 12 (23), 3421-3424.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
