4-Azaindole

4-Azaindole is a scaffold. 4-Azaindole can be used in the synthesis of Nav1.2 inhibitors. 4-Azaindole can be used in epilepsy and breast cancer research[1][2].

Product Specifications

CAS Number

[272-49-1]

UNSPSC

12352200

Hazard Statement

H302, H315, H319, H335

Target

Biochemical Assay Reagents; Drug Intermediate

Type

Biochemical Assay Reagents

Related Pathways

Others

Field of Research

Cancer; Neurological Disease

Assay Protocol

https://www.medchemexpress.com/4-azaindole.html

Purity

99.57

Solubility

10 mM in DMSO

Smiles

C12=NC=CC=C1NC=C2

Molecular Formula

C7H6N2

Molecular Weight

118.14

Precautions

H302, H315, H319, H335

References & Citations

[1]Lou B, et al. Discovery of novel 4-azaindole derivatives as selective Nav1.2 Inhibitor with potent antiepileptic activity and low neurotoxicity. Eur J Med Chem. 2025 Aug 5;292:117664. |[2]Venkat Swamy P, et al. Amide derivatives of 4-azaindole: Design, synthesis, and EGFR targeting anticancer agents. Synthetic Communications, 2020, 50 (1) : 71-84.