Ubavitinib (tosylate)
AZD3229 Tosylate is a potent pan-KIT mutant inhibitor for the treatment of gastrointestinal stromal tumors.
Product Specifications
CAS Number
[2248003-71-4]
Product Name Alternative
AZD3229 (tosylate)
UNSPSC
12352005
Target
C-Kit
Type
Reference compound
Related Pathways
Protein Tyrosine Kinase/RTK
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/AZD3229_Tosylate.html
Purity
98.83
Solubility
DMSO : ≥ 100 mg/mL
Smiles
COCCOC1=CC(F)=C2C(N=CN=C2NC3=CC=C(NC(CN4C=C(C(C)C)N=N4)=O)C=C3)=C1.CC5=CC=C(S(O)(=O)=O)C=C5
Molecular Formula
C31H34FN7O6S
Molecular Weight
651.71
References & Citations
[1]Kettle JG, et al. Discovery of N- (4-{[5-Fluoro-7- (2-methoxyethoxy) quinazolin-4-yl]amino}phenyl) -2-[4- (propan-2-yl) -1 H-1,2,3-triazol-1-yl]acetamide (AZD3229), a Potent Pan-KIT Mutant Inhibitor for the Treatment of Gastrointestinal Stromal Tumors. J Med Chem. 2018 Oct 11;61 (19) :8797-8810.
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Curated Selection
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