PD 165929
PD 165929 is a high affinity and competitive non-peptide neuromedin-B (NMB) receptor selective antagonist (Ki: 6.3 nM; IC50: 150 nM for rat NMB receptor) [1].
Product Specifications
CAS Number
185215-75-2
UNSPSC
12352005
Target
Bombesin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Smiles
CC(C)C(C=CC=C1C(C)C)=C1NC(N[C@](CC2=CNC3=CC=CC=C23)(C)C(NCC4(C5=CC=CC=N5)CCCCC4)=O)=O
Molecular Formula
C37H47N5O2
Molecular Weight
593.80
References & Citations
[1]J.M. Eden, et al. PD 165929 -the first high affinity non-peptide neuromedin-B (NMB) receptor selective antagonist. Bioorganic & Medicinal Chemistry Letters. Volume 6, Issue 21
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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