Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

CCR2 antagonist 1

CCR2 antagonist 1 (compound 15a) is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM[1].

Product Specifications

CAS Number

1683534-96-4

UNSPSC

12352005

Hazard Statement

H315-H319-H320

Target

CCR

Type

Reference compound

Related Pathways

GPCR/G Protein; Immunology/Inflammation

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/CCR2_antagonist_1.html

Purity

98.00

Solubility

DMSO : 125 mg/mL (ultrasonic)

Smiles

O=C([C@]1(C(C)C)C[C@H](N[C@@H]2CCC3=C2C=CC(Br)=C3)CC1)N4CC5=C(C=CC(C(F)(F)F)=C5)CC4

Molecular Formula

C28H32BrF3N2O

Molecular Weight

549.47

Precautions

P264-P280-P302+P352-P305+P351+P338-P362

References & Citations

[1]Vilums M, et al. When structure-affinity relationships meet structure-kinetics relationships: 3- ((Inden-1-yl) amino) -1-isopropyl-cyclopentane-1-carboxamides as CCR2 antagonists. Eur J Med Chem. 2015 Mar 26;93:121-34.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

CCR2

Available Sizes

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

6xHistidine Epitope Tag (HHHHHH) Mouse Monoclonal Antibody [Clone ID: 16-002]
AM26098PU-N 100 µg

6xHistidine Epitope Tag (HHHHHH) Mouse Monoclonal Antibody [Clone ID: 16-002]

Sign In for Pricing
View Details
CD32A (FCGR2A) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI6D11]
TA500653AM 100 µL

CD32A (FCGR2A) Mouse Monoclonal Antibody (Biotin conjugated) [Clone ID: OTI6D11]

Sign In for Pricing
View Details
IGHM Mouse Monoclonal Antibody [Clone ID: 3E12-H4-G4]
TA384502 100 µL

IGHM Mouse Monoclonal Antibody [Clone ID: 3E12-H4-G4]

Sign In for Pricing
View Details
XFD594-Wheat Germ Agglutinin (WGA) Conjugate
25509-AAT 1 mg

XFD594-Wheat Germ Agglutinin (WGA) Conjugate

Sign In for Pricing
View Details
RPS27A (NM_002954) Human Over-expression Lysate
LC401036 20 µg

RPS27A (NM_002954) Human Over-expression Lysate

Sign In for Pricing
View Details
Human LUZP2 activation kit by CRISPRa
GA117377 1 Kit

Human LUZP2 activation kit by CRISPRa

Sign In for Pricing
View Details