K- (D-1-Nal) -FwLL-NH2
K- (D-1-Nal) -FwLL-NH2 is a high affinity, potent and inverse ghrelin receptor agonist (EC50=3.4 nM, Ki=4.9 nM) . K- (D-1-Nal) -FwLL-NH2 can be used for the research of obesity[1].
Product Specifications
CAS Number
1394288-22-2
UNSPSC
12352209
Target
GHSR
Type
Peptides
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/k-d-1-nal-fwll-nh2.html
Solubility
10 mM in DMSO
Smiles
CC(C)C[C@@H](C(N)=O)NC([C@H](CC(C)C)NC([C@@H](CC1=CNC2=C1C=CC=C2)NC([C@H](CC3=CC=CC=C3)NC([C@@H](CC4=C5C=CC=CC5=CC=C4)NC([C@H](CCCCN)N)=O)=O)=O)=O)=O
Molecular Formula
C51H67N9O6
Molecular Weight
902.13
References & Citations
[1]Els S, et al. An aromatic region to induce a switch between agonism and inverse agonism at the ghrelin receptor. J Med Chem. 2012;55 (17) :7437-7449.
Shipping Conditions
Room temperature
Scientific Category
Peptides
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
