GSK1104252A
GSK1104252A is a potent and selective GPR119 agonist. GSK1104252A can be used for type 2 diabetes research[1].
Product Specifications
CAS Number
1001397-20-1
UNSPSC
12352005
Target
GPR119
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gsk1104252a.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCC(OC2=C3C(N(C4=CC=C(S(=O)(C)=O)C=C4F)CC3)=NC=N2)CC1)OC(C)C
Molecular Formula
C22H27FN4O5S
Molecular Weight
478.54
References & Citations
[1]Subba R Katamreddy, et al. Discovery of 6,7-dihydro-5H-pyrrolo[2,3-a]pyrimidines as orally available G protein-coupled receptor 119 agonists. J Med Chem. 2012 Dec 27;55 (24) :10972-94.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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