SSTR5 antagonist 6
SSTR5 antagonist 6 is an orally active somatostatin receptor subtype 5 (SSTR5) antagonist with an IC50 of 24 nM. SSTR5 antagonist 6 can be used in the study of type 2 diabetes[1].
Product Specifications
CAS Number
1007836-12-5
UNSPSC
12352005
Target
Somatostatin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/sstr5-antagonist-6.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CN=C(NC2CCN(CC2)CC3=CC(OCC)=C(C(OCC)=C3)Cl)C=C1)O
Molecular Formula
C22H28ClN3O4
Molecular Weight
433.93
References & Citations
[1]Sprecher, Urs et al. Novel, non-peptidic somatostatin receptor subtype 5 antagonists improve glucose tolerance in rodents. Regulatory peptides vol. 159,1-3 (2010) : 19-27.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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