GPR132 antagonist 1 (dihydrocholide)
GPR132 antagonist 1 dihydrocholide (GPR132-B-160, Compound 25) is a GPR132 antagonist with an EC50 value of 0.075 μM. GPR132 antagonist 1 dihydrocholide has promote insulin secretion activity with an EC50 value of 0.7 μM[1].
Product Specifications
UNSPSC
12352005
Target
G2A (GPR132)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/gpr132-antagonist-1-dihydrocholide.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=C(C)C2=C(C=CC(S(=O)(NCCC3=CC=CC=C3)=O)=C2)O1)O.[H]Cl.[H]Cl
Molecular Formula
C18H19Cl2NO5S
Molecular Weight
432.32
References & Citations
[1]Ning Jiao, et al. GPCR modulators and uses thereof. CN116903563A.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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