DPI-287
DPI-287 is a selective delta-opioid receptor (DOP) agonist with a Ki value of 0.39 nM and can be used for pain research[1].
Product Specifications
CAS Number
519058-13-0
UNSPSC
12352005
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/dpi-287.html
Solubility
10 mM in DMSO
Smiles
C[C@@H](CN([C@@H](C1)C)CC2=CC=CC=C2)N1[C@@H](C3=CC(O)=CC=C3)C4=CC=C(C=C4)C(N(CC)CC)=O
Molecular Formula
C31H39N3O2
Molecular Weight
485.66
References & Citations
[1]Claff T, et al. Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists. Sci Adv. 2019 Nov 27;5 (11) :eaax9115.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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