RXFP1 receptor agonist-8
RXFP1 receptor agonist-8 (Example 2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-8 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.8 nM[1].
Product Specifications
CAS Number
[2941271-76-5]
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-8.html
Solubility
10 mM in DMSO
Smiles
O=C(NC1=C(C(NC2=CC=C(F)C(C(F)(F)F)=C2)=O)C=C(CCCC3)C3=C1)C4=CC(C5=C(F)C=CC(C(C(O)=O)NC(C6CCOCC6)=O)=C5)=CC=C4OC
Molecular Formula
C40H36F5N3O7
Molecular Weight
765.72
References & Citations
[1]Jones, Clifford D., et al. Prepration of pyridopyrimidines as KRAS mutant proteins inhibitors useful in treatment of cancers. Patent. WO2022248885.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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