RXFP1 receptor agonist-5
RXFP1 receptor agonist-5 (Example 98) is a RXFP1 receptor agonist. RXFP1 receptor agonist-5 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1.3 nM[1].
Product Specifications
CAS Number
2941385-36-8
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-5.html
Solubility
10 mM in DMSO
Smiles
OCC1C[C@@]2([H])C(C3=CC(C(NC4=C(C=C5C(OC(F)(O5)F)=C4)C(NC6=CC(C(F)(F)F)=C(C=C6)F)=O)=O)=C(C=C3)OC)=NO[C@@]2([H])C1
Molecular Formula
C30H23F6N3O7
Molecular Weight
651.51
References & Citations
[1]Sreekantha Ratna KUMAR, et al. Benzothiazole, benzoisoxazole and benzodioxole analogs as rxfp1 receptor agonists. Patent. WO2023114822A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
Explore Other Products
Browse additional items from our catalog
ACTH (Adrenocorticotrophic Hormone) (AH26), CF594 conjugate, 0.1mg/mL
Cytokeratin 8/18 (C-51), CF640R conjugate, 0.1mg/mL
ACTH (Adrenocorticotrophic Hormone) (AH26), CF740 conjugate, 0.1mg/mL
