RXFP1 receptor agonist-4
RXFP1 receptor agonist-4 (Example 268) is a RXFP1 receptor agonist. RXFP1 receptor agonist-4 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 4.9 nM[1].
Product Specifications
CAS Number
2941376-76-5
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-4.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC(C2=NOC3C2CC(CO)C3)=CC=C1OC)NC4=C(C(NC5=CC=C(F)C(C(F)(F)F)=C5)=O)SC6=CC(C(F)(F)F)=CC=C64
Molecular Formula
C32H24F7N3O5S
Molecular Weight
695.60
References & Citations
[1]Sreekantha Ratna KUMAR, et al. Benzothiophene derivatives as rxfp1 agonists. Patent. WO2023114823A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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