RXFP1 receptor agonist-3
RXFP1 receptor agonist-3 (Example 223) is a RXFP1 receptor agonist. RXFP1 receptor agonist-3 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 2 nM[1].
Product Specifications
CAS Number
2924767-53-1
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-3.html
Solubility
10 mM in DMSO
Smiles
O=C(N[C@@H]1[C@@H]2CC[C@@H](/C2=C/C3CC3)[C@@H]1C(NC4=CC(C(F)(F)F)=C(F)C=C4)=O)C5=CC(C6=C(F)C=CC(C(OC(NC7=CC=CC=C7F)=O)C(F)(F)F)=C6)=CC=C5OC
Molecular Formula
C42H34F9N3O5
Molecular Weight
831.72
References & Citations
[1]Shun Su, et al. Rxfp1 agonists. Patent. WO2023076626A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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