RXFP1 receptor agonist-2

RXFP1 receptor agonist-2 (Example 124) is a RXFP1 receptor agonist. RXFP1 receptor agonist-2 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1 nM[1].

Product Specifications

CAS Number

[2924460-54-6]

UNSPSC

12352005

Target

RXFP Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

COVID-19-immunoregulation

Field of Research

Inflammation/Immunology; Cardiovascular Disease

Assay Protocol

https://www.medchemexpress.com/rxfp1-receptor-agonist-2.html

Solubility

10 mM in DMSO

Smiles

O=C(N1CCC(O)CC1)/C=C/C2=CC=C(OC)C(C(N[C@@H]3[C@@H]4CC[C@@H](/C4=C/C(F)(F)F)[C@@H]3C(NC5=CC(C(F)(F)F)=C(F)C=C5)=O)=O)=C2

Molecular Formula

C33H32F7N3O5

Molecular Weight

683.61

References & Citations

[1]Scott A. SHAW, et al. Rxfp1 agonists. Patent. WO2023077040.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

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