RXFP1 receptor agonist-2
RXFP1 receptor agonist-2 (Example 124) is a RXFP1 receptor agonist. RXFP1 receptor agonist-2 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1 nM[1].
Product Specifications
CAS Number
[2924460-54-6]
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-2.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCC(O)CC1)/C=C/C2=CC=C(OC)C(C(N[C@@H]3[C@@H]4CC[C@@H](/C4=C/C(F)(F)F)[C@@H]3C(NC5=CC(C(F)(F)F)=C(F)C=C5)=O)=O)=C2
Molecular Formula
C33H32F7N3O5
Molecular Weight
683.61
References & Citations
[1]Scott A. SHAW, et al. Rxfp1 agonists. Patent. WO2023077040.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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