RXFP1 receptor agonist-2
RXFP1 receptor agonist-2 (Example 124) is a RXFP1 receptor agonist. RXFP1 receptor agonist-2 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 1 nM[1].
Product Specifications
CAS Number
[2924460-54-6]
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-2.html
Solubility
10 mM in DMSO
Smiles
O=C(N1CCC(O)CC1)/C=C/C2=CC=C(OC)C(C(N[C@@H]3[C@@H]4CC[C@@H](/C4=C/C(F)(F)F)[C@@H]3C(NC5=CC(C(F)(F)F)=C(F)C=C5)=O)=O)=C2
Molecular Formula
C33H32F7N3O5
Molecular Weight
683.61
References & Citations
[1]Scott A. SHAW, et al. Rxfp1 agonists. Patent. WO2023077040.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
More Discoveries
Explore Other Products
Browse additional items from our catalog
MBS9350667 Inquire
Chicken Killer Cell Lectin Like Receptor Subfamily A, Member 1 (KLRA1) ELISA Kit
Sign In for Pricing
View Details 
302273-ML550 100 µL
ARL6 (ADP-Ribosylation Factor-like Protein 6, Bardet-Biedl Syndrome 3 Protein, ARL6, BBS3) (MaxLight 550) discontinued
Sign In for Pricing
View Details K1144403 1.0 µg DNA
KIAA1881 sgRNA CRISPR Lentivector (Human) (Target 2)
Sign In for Pricing
View Details