RXFP1 receptor agonist-1
RXFP1 receptor agonist-1 (Example 2 peak2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-1 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 300 nM[1].
Product Specifications
CAS Number
[2924619-64-5]
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-1.html
Solubility
10 mM in DMSO
Smiles
O=C(N[C@@H]1[C@@H]2CC[C@@H](/C2=C/C(F)(F)F)[C@@H]1C(NC3=CC(C(F)(F)F)=C(F)C=C3)=O)[C@@H](C4)CCC[C@@H]4C5=CC(C(O)=O)=CC=C5
Molecular Formula
C31H29F7N2O4
Molecular Weight
626.56
References & Citations
[1]Donald J.P. Pinto, et al. Rxfp1 modulators for the treatment of heart failure. Patent. WO2023077041A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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