RXFP1 receptor agonist-1
RXFP1 receptor agonist-1 (Example 2 peak2) is a RXFP1 receptor agonist. RXFP1 receptor agonist-1 stimulates cAMP production in HEK293 cells stably expressing human RXFP1, with an EC50 value of 300 nM[1].
Product Specifications
CAS Number
[2924619-64-5]
UNSPSC
12352005
Target
RXFP Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rxfp1-receptor-agonist-1.html
Solubility
10 mM in DMSO
Smiles
O=C(N[C@@H]1[C@@H]2CC[C@@H](/C2=C/C(F)(F)F)[C@@H]1C(NC3=CC(C(F)(F)F)=C(F)C=C3)=O)[C@@H](C4)CCC[C@@H]4C5=CC(C(O)=O)=CC=C5
Molecular Formula
C31H29F7N2O4
Molecular Weight
626.56
References & Citations
[1]Donald J.P. Pinto, et al. Rxfp1 modulators for the treatment of heart failure. Patent. WO2023077041A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Explore Other Products
Browse additional items from our catalog
Actin filament-associated protein 1 (AFAP1) Chicken ELISA Kit