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CRF1 receptor antagonist-1

Product Specifications

UNSPSC Description

CRF1 receptor antagonist-1 (Compound 2) is a CRF1 receptor antagonist. CRF1 receptor antagonist-1 can be used for research of congenital adrenal hyperplasia (CAH)[1].

Target Antigen

CFTR

Type

Reference compound

Related Pathways

Membrane Transporter/Ion Channel

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Endocrinology

Assay Protocol

https://www.medchemexpress.com/crf1-receptor-antagonist-1.html

Solubility

10 mM in DMSO

Smiles

C#CCN(C1=NC(C2=C(C=C(C(C)=C2)OC)Cl)=C(S1)C)[C@H](C3=CC(F)=C(C=C3)CO)CC4CC4

Molecular Weight

499.04

References & Citations

[1]Evan Smith, et al. Crf receptor antagonists and methods of use. Patent. WO2021062246.

Shipping Conditions

Room temperature

Product Datasheet

http://file.medchemexpress.com/batch_PDF/HY-156522/CRF1-receptor-antagonist-1-DataSheet-MedChemExpress.pdf

Product MSDS

http://file.medchemexpress.com/batch_PDF/HY-156522/

Clinical Information

No Development Reported

CAS Number

2635364-30-4

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