CB2 receptor antagonist 4
Product Specifications
UNSPSC Description
CB2 receptor antagonist 4 (compound (R)-1) is a CB2R-selective inverse agonist with a Kd value of 39 nM[1].
Target Antigen
Others
Type
Reference compound
Related Pathways
Others
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb2-receptor-antagonist-4.html
Solubility
10 mM in DMSO
Smiles
CC(C1=CC(OC)=C([C@@]2([H])C=C(CN)[C@@H]3C(C)(C)[C@H]2C3)C(OC)=C1)(C)[C@H](CCCCCN=[N+]=[N-])C4=CC=CC=C4
Molecular Weight
530.74
References & Citations
[1]Erick Carreira, et al. Flipping the GPCR Switch: Structure–Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists. ChemRxiv. 2023.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-155481A/CB2-receptor-antagonist-4-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-155481A/
Clinical Information
No Development Reported
Curated Selection
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