CB2 receptor antagonist 4
CB2 receptor antagonist 4 (compound (R) -1) is a CB2R-selective inverse agonist with a Kd value of 39 nM[1].
Product Specifications
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb2-receptor-antagonist-4.html
Solubility
10 mM in DMSO
Smiles
CC(C1=CC(OC)=C([C@@]2([H])C=C(CN)[C@@H]3C(C)(C)[C@H]2C3)C(OC)=C1)(C)[C@H](CCCCCN=[N+]=[N-])C4=CC=CC=C4
Molecular Formula
C33H46N4O2
Molecular Weight
530.74
References & Citations
[1]Erick Carreira, et al. Flipping the GPCR Switch: Structure–Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists. ChemRxiv. 2023.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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