Besipirdine
Besipirdine is a non-receptor-dependent cholinomimetic agent with noradrenergic activity. Besipirdine inhibits voltage-dependent sodium and potassium channels.
Product Specifications
CAS Number
119257-34-0
Product Name Alternative
HP 749 (free base)
UNSPSC
12352005
Target
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/besipirdine.html
Solubility
10 mM in DMSO
Smiles
CCCN(C1=CC=NC=C1)N2C=CC3=C2C=CC=C3
Molecular Formula
C16H17N3
Molecular Weight
251.33
References & Citations
[1]Hsu RS, DiLeo EM, Chesson SM, Klein JT, Effland RC. Determination of HP 749, a potential therapeutic agent for Alzheimer's disease, in plasma by high-performance liquid chromatography. J Chromatogr. 1991;572 (1-2) :352-359. |[2]Tang L, Smith CP, Huger FP, Kongsamut S. Effects of besipirdine at the voltage-dependent sodium channel. Br J Pharmacol. 1995;116 (5) :2468-2472.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 3
Available Sizes
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