AP-C2

AP-C2 is a potent guanosine 3',5'-cyclic monophosphate (cGMP) -dependent protein kinase II (cGKII) inhibitor with a pIC50 of 5.2[1].

Product Specifications

CAS Number

[682793-07-3]

UNSPSC

12352005

Target

Ser/Thr Protease

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Metabolism-protein/nucleotide metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/ap-c2.html

Solubility

10 mM in DMSO

Smiles

C1(C2=CC=CS2)=CC=NC(NCCC3=CNC4=C3C=CC=C4)=N1

Molecular Formula

C18H16N4S

Molecular Weight

320.41

References & Citations

[1]Marcel J C Bijvelds, et al. Selective inhibition of intestinal guanosine 3',5'-cyclic monophosphate signaling by small-molecule protein kinase inhibitors. J Biol Chem. 2018 May 25;293 (21) :8173-8181.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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