DRAK1/2-IN-1
DRAK1/2-IN-1 (compound 10e) is an active dual DRAK1 and DRAK2 inhibitor with Kd values of 1 μM and 6 μM, respectively[1].
Product Specifications
CAS Number
1629227-34-4
UNSPSC
12352005
Target
DAPK
Type
Reference compound
Related Pathways
Apoptosis
Applications
COVID-19-immunoregulation
Field of Research
Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/drak1-2-in-1.html
Solubility
10 mM in DMSO
Smiles
O=C(C1CCCCC1)NC2=CSC3=NC=C(C4=CC(OC)=C(OC)C=C4)C=C32
Molecular Formula
C22H24N2O3S
Molecular Weight
396.50
References & Citations
[1]Gao LJ, et al. Discovery of dual death-associated protein related apoptosis inducing protein kinase 1 and 2 inhibitors by a scaffold hopping approach. J Med Chem. 2014 Sep 25;57 (18) :7624-43.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog