Tankyrase-IN-3
Tankyrase-IN-3 is a tankyrase 1 (TNKS1) inhibitor with an IC50 value of 22 nM. Tankyrase-IN-3 can be used for the research of cancer[1].
Product Specifications
CAS Number
938893-79-9
UNSPSC
12352005
Target
PARP
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage; Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/tankyrase-in-3.html
Solubility
10 mM in DMSO
Smiles
O=C(OCC(N1CCN(CC1)C2=CC=CC=N2)=O)CC(C3=CC=CC=C34)=NNC4=O
Molecular Formula
C21H21N5O4
Molecular Weight
407.42
References & Citations
[1]Alba L Montoya, et al. Combining pharmacophore models derived from DNA-encoded chemical libraries with structure-based exploration to predict Tankyrase 1 inhibitors. Eur J Med Chem. 2023 Jan 15;246:114980.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
TNKS1/PARP5A
Frequently Asked Questions
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