CYP1B1-IN-5

CYP1B1-IN-5 (Compound 6q) is a potent and selective cytochrome P450 1B1 (CYP1B1) inhibitor with an IC50 of 4.7 nM[1].

Product Specifications

CAS Number

[176442-56-1]

UNSPSC

12352005

Target

Cytochrome P450

Type

Reference compound

Related Pathways

Metabolic Enzyme/Protease

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/cyp1b1-in-5.html

Purity

98.03

Solubility

DMSO : 20 mg/mL (ultrasonic; warming; heat to 60°C)

Smiles

O=C1OC(C2=CC=C(C=C2)I)=NC3=C1C=CC=C3

Molecular Formula

C14H8INO2

Molecular Weight

349.12

References & Citations

[1]Yi L, et al. A new class of CYP1B1 inhibitors derived from bentranil. Bioorg Med Chem Lett. 2022 Dec 21;80:129112.

Shipping Conditions

Room Temperature

Storage Conditions

-20°C, 3 years; 4°C, 2 years (Powder)

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

CYP1

Available Sizes

Curated Selection

Explore Other Products

Discover premium biology products from our extensive collection of 20M+ items

FAB10866CL1 0.1 mL

Mouse Monoclonal PD-1 Antibody (1026519) [CoraFluor 1]

Ask

View Details

7300 15 x 11 x 4 cm

Drug Powders, 25 microscope slides

Ask

View Details

MBS8421921-01 0.12 mL

Rabbit Anti Human LAMA1 Polyclonal Affinity Purified (PBS with 0.05% sodium azide and 50% glycerol, pH7.4)(IHC, ELISA)

Ask

View Details

MBS8421921-02 0.2 mL

Rabbit Anti Human LAMA1 Polyclonal Affinity Purified (PBS with 0.05% sodium azide and 50% glycerol, pH7.4)(IHC, ELISA)

Ask

View Details

MBS8421921-03 5x 0.2 mL

Rabbit Anti Human LAMA1 Polyclonal Affinity Purified (PBS with 0.05% sodium azide and 50% glycerol, pH7.4)(IHC, ELISA)

Ask

View Details

APR23502N-01 50 µL

KEAP1 Rabbit pAb (APR23502N)

Ask

View Details