ChoKα inhibitor-5
ChoKα inhibitor-5 is a sulphur-containing choline kinase inhibitor. ChoKα inhibitor-5 can inhibit HChoK α1 with an IC50 value of 0.64 μM. ChoKα inhibitor-5 also can induce apoptosis. ChoKα inhibitor-5 can be used for the research of cancer[1].
Product Specifications
UNSPSC
12352005
Target
Apoptosis
Type
Reference compound
Related Pathways
Apoptosis
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/chokα-inhibitor-5.html
Solubility
10 mM in DMSO
Smiles
C=CCCCCN(C1=CC=[N+](C2=C1SC=C2)CC3=CC=C(C=C3)SCCSC4=CC=C(C=C4)C[N+]5=CC=C(C6=C5C=CS6)N(CCCCC=C)CCCCC=C)CCCCC=C.[Br-].[Br-]
Molecular Formula
C54H68Br2N4S4
Molecular Weight
1061.21
References & Citations
[1]Pilar M Luque-Navarro, et al. New bioisosteric sulphur-containing choline kinase inhibitors with a tracked mode of action. Eur J Med Chem. 2023 Jan 15;246:115003.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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