Anticancer agent 84

Anticancer agent 84 is an anticancer agent. Anticancer agent 84 represses the transcription of c-MYC by stabilizing the G-quadruplex (G4) structure. Anticancer agent 84 can be used for the research of cancer[1].

Product Specifications

CAS Number

[2714510-72-0]

UNSPSC

12352005

Target

C-Myc

Type

Reference compound

Related Pathways

Apoptosis

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/anticancer-agent-84.html

Solubility

10 mM in DMSO

Smiles

CCN1C2=CC=C(C=C2C3=C1C=CC=C3)C4=NC(C5=CC=C(C=C5)N6CCN(CC6)C)=C(N4C7=CC=C(C=C7)OCCOCCOC8(O[C@@H]9O[C@H]([C@@H]([C@H]([C@@H]9O8)O)O)CO)C)C%10=CC=C(C=C%10)N%11CCN(CC%11)C

Molecular Formula

C57H67N7O9

Molecular Weight

994.18

References & Citations

[1]Mao-Lin Li, et al. Design, Synthesis, and Evaluation of New Sugar-Substituted Imidazole Derivatives as Selective c-MYC Transcription Repressors Targeting the Promoter G-Quadruplex. J Med Chem. 2022 Sep 19.