RS6212
RS6212 is a specific LDH (lactate dehydrogenase) inhibitor with an IC50 value of 12.03 μM . RS6212 inhibits tumor growth and exhibits potent anticancer activity in multiple cancer cell lines[1].
Product Specifications
CAS Number
2097925-52-3
UNSPSC
12352005
Target
Lactate Dehydrogenase; Oxidative Phosphorylation
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/rs6212.html
Purity
98.86
Solubility
DMSO : 16.67 mg/mL (ultrasonic; warming; heat to 60°C)
Smiles
O=C1C=C(CCC2)C2=NN1CC3CCN(C(C4=CC=CC=C45)=NS5(=O)=O)CC3
Molecular Formula
C20H22N4O3S
Molecular Weight
398.48
References & Citations
[1]Di Magno L, et al. Discovery of novel human lactate dehydrogenase inhibitors: Structure-based virtual screening studies and biological assessment. Eur J Med Chem. 2022 Jul 14. 240:114605.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
TP322932 20 µg
Neuroligin 4 (NLGN4X) (NM_020742) Human Recombinant Protein
Sign In for Pricing
View Details ![LDHB Mouse Monoclonal Antibody [Clone ID: AT14D7]](https://cdn.genprice.uk/products/937/68dd189e061270361e8fd933/imageurl/am50625pu-s.webp)
AM50625PU-S 50 µL
LDHB Mouse Monoclonal Antibody [Clone ID: AT14D7]
Sign In for Pricing
View Details