ER degrader 4

ER degrader 4 is a selective and orally active estrogen receptor degrader. ER degrader 4 has anti-tumor activity[1].

Product Specifications

CAS Number

[2913192-39-7]

UNSPSC

12352005

Target

Estrogen Receptor/ERR

Type

Reference compound

Related Pathways

Vitamin D Related/Nuclear Receptor

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/er-degrader-4.html

Solubility

10 mM in DMSO

Smiles

O=C(C1=C(C=C(C=C1)C)C)C(SC2=CC(F)=CC=C23)=C3OC4=CC=C(C=C4)/C=C/C(O)=O

Molecular Formula

C26H19FO4S

Molecular Weight

446.49

References & Citations

[1]Lu Y, et al. Design, synthesis and biological evaluation of fluorinated selective estrogen receptor degraders (FSERDs) --- A promising strategy for advanced ER positive breast cancer. Eur J Med Chem. 2023 May 5;253:115324.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Curated Selection

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