GSK023
GSK023 (compound 31) is a selective chemical probe targeting the BET BD1 domain[1].
Product Specifications
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/gsk023.html
Solubility
10 mM in DMSO
Smiles
O=C1C(C)=CC(C2=NC3=CC=CC=C3N2C[C@H]4CN(C(C5CCN(C(C)C)CC5)=O)CCC4)=CN1C
Molecular Formula
C29H39N5O2
Molecular Weight
489.65
References & Citations
[1]Bradley E et al. Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N-Terminal Bromodomain Chemical Probe. J Med Chem. 2023 Nov 15.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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